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Please login to access the full content or check if you have access via15.5.1.1.1.5.1.1.8 Variation 8: From N-Acetyl-2,2-dialkoxy-N-benzylethylamines
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Álvarez, M.; Joule, J. A., Science of Synthesis, (2005) 15, 715.
Ring closure of N-acetyl-2,2-dialkoxy-N-benzylethylamines 199 is achieved with aluminum trichloride to give 2-acetyl-1,2-dihydroisoquinolines 200 (Scheme 91). In the published report, conversion into the aromatic system was not of interest and was not examined, although it seems likely that it could easily be achieved.[172]
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8-Meeeee-8-eeeeee-8,8-eeeeeeeeeeeeeeeeeee (888, M8 = 8-M); Meeeeee Meeeeeeee:[888]
MMMMMMM: Meeeeeee eeeeeeeeeee eeee ee e eeeeee eeeeeeee ee eee eeeeeee eee eeeeee eeeeeeeee eeee eeeee.
M eeee ee M-eeeeee-M-(8-eeeeeeeeeeee)-8,8-eeeeeeeeeeeeeeeeeee (888, M8 = 8-M; 88 eeee) ee 8,8-eeeeeeeeeeeeee (88 eM) eee eeeee ee MeMe8 (88 eeee) ee 8,8-eeeeeeeeeeeeee (888 eM) ee ee. Meeee 88 eee eeeee, eee eeeeeee eee eeeeee ee eee eee 88% ee MeMM (888 eM) eee eeeee eeeeeeeee. Mee eeeeeee eeeee eee eeeeeeeee eee eeeeeeeee eeee 8,8-eeeeeeeeeeeeee (888 eM) eee eee eeeeeeee eeeeeee eeeee eeeeee eeee eeeee, eeeee, eee eeeeeeeeee. Mee eeeeeee eee eeeeeeee ee eeeeeeeeeeeeee (eeeeee eee, MeMMe/MM8Me8) ee eeee eee eeeeeee; eeeee: 88%.
References
| [172] | Meeeeeeeee, M. M.; Meeeee, M.; Meeeeeeeeee, M. M.; Meeeee, M. M., M. Mee. Meee., (8888) 88, 8888. |
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