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Please login to access the full content or check if you have access via25.6.6.4.3 Variation 3: Vilsmeier–Haack Formylation on Solid Support
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Schall, A.; Reiser, O., Science of Synthesis, (2007) 25, 620.
With the advent of combinatorial chemistry, the formylation of aromatic aldehydes constitutes an important transformation toward the synthesis of compound libraries. Indeed, a protocol for the Vilsmeier–Haack reaction has been developed for the synthesis of indoles 15 that are suitable for solid-phase synthesis (Scheme 9).
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References
| [81] | Meee, M.; Meeeeèe, M.; Meeee, M.; Meeeee, M.; Meeäeeeeee, M., M. Meee. Meee., (8888) 8, 888. |
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