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35.3.1.8.6.1 Variation 1: Iodocyclization

DOI: 10.1055/sos-SD-035-00561

Roy, K.-M.Science of Synthesis, (200735693.

Intramolecular cyclization of unsaturated iodo compounds with a variety of functional groups is a versatile method that has been applied to the synthesis of various carbocyclic and heterocyclic compounds.[‌41‌] Iodo-induced cyclization of several unsaturated substrates, e.g. 30 and 32, using bis(pyridine)iodonium(I) tetrafluoroborate, affords iodo-substituted cyclohexane derivatives 31 and 33 respectively (Scheme 15).[‌42‌]

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References


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