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Please login to access the full content or check if you have access via Variation 3: Cyclization of 2-Azidoalkanols

DOI: 10.1055/sos-SD-040-00445

Sweeney, J. B.Science of Synthesis, (200940698.

The conversion of 2-azidoalkanols into aziridines using phosphines was first reported in 1978 (Scheme 114),[‌313‌] since when the method has frequently been exploited to enable the synthesis of aziridines such as 196.[‌314‌‌316‌]

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