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DOI: 10.1055/sos-SD-110-00001

Joule, J. A.Science of Synthesis Knowledge Updates, (2010264.

A range of 2-aryl-1H-indoles 226 can be prepared (Scheme 80) from 2,2,2-trifluoro-N-(2-iodophenyl)acetamide using various copper catalysts, the best of which is (1,10-phenanthroline)bis(triphenylphosphine)copper(I) nitrate [Cu(phen)(PPh3)2]NO3, used in the presence of potassium phosphate.[‌257‌]

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