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DOI: 10.1055/sos-SD-208-00030

Scholz, U.; Dong, W.; Feng, J.; Shi, W.Science of Synthesis: Cross Coupling and Heck-Type Reactions, (20132102.

The scope of the nickel–phenanthroline–polymethylhydrosiloxane catalytic system can also be extended to 2-chloroquinoline.[‌102‌,‌108‌] The amination of 2-chloroquinoline with either pyrrolidine or 4,4-dimethoxypiperidine gives the desired products 88 in excellent yields (Scheme 61).[‌108‌]

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