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DOI: 10.1055/sos-SD-110-00001

Joule, J. A.Science of Synthesis Knowledge Updates, (2010263.

Conducting the Larock synthesis in the presence of an aryl halide allows the trapping of the intermediate organopalladium intermediate and thus the linking of that aromatic moiety to the forming indole 3-position to give 225 (Scheme 79).[‌256‌]

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